Development of Oxygen-Bridged Pyrazole-Based Structures as Cannabinoid Receptor 1 Ligands
In this work, the synthesis of the cannabinoid receptor 1 neutral antagonists 8-chloro-1-(2,4-dichlorophenyl)-<i>N</i>-piperidin-1-yl-4,5-dihydrobenzo-1<i>H</i>-6-oxa-cyclohepta[1,2-<i>c</i>]pyrazole-3-carboxamide <b>1a</b> and its deaza <i>N-<...
Main Authors: | Gabriele Murineddu, Battistina Asproni, Paola Corona, Sandra Piras, Paolo Lazzari, Stefania Ruiu, Laura Legnani, Lucio Toma, Gérard A. Pinna |
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Format: | Article |
Language: | English |
Published: |
MDPI AG
2019-04-01
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Series: | Molecules |
Subjects: | |
Online Access: | https://www.mdpi.com/1420-3049/24/9/1656 |
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