Search Results - Marcelo A. Comini
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Glucose 6-Phosphate Dehydrogenase from Trypanosomes: Selectivity for Steroids and Chemical Validation in Bloodstream <i>Trypanosoma brucei</i> by Cecilia Ortíz, Francesca Moraca, Marc Laverriere, Allan Jordan, Niall Hamilton, Marcelo A. Comini
Published in Molecules (2021-01-01)Get full text
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Diglycosyl diselenides alter redox homeostasis and glucose consumption of infective African trypanosomes by Jaime Franco, Florencia Sardi, László Szilágyi, Katalin E. Kövér, Krisztina Fehér, Marcelo A. Comini
Published in International Journal for Parasitology: Drugs and Drug Resistance (2017-12-01)Get full text
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Expression and functional characterization of chimeric recombinant bovine follicle‐stimulating hormone produced in Leishmania tarentolae by Cecilia Abreu, Karin Grunberg, Mariana Bonilla, Martina Crispo, Sergio Pantano, Julian Jaeschke, Marcelo A. Comini, Mariela Bollati‐Fogolín
Published in Microbial Biotechnology (2024-04-01)Get full text
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Evaluation of the Anti-<i>Leishmania mexicana</i> and -<i>Trypanosoma brucei</i> Activity and Mode of Action of 4,4′-(Arylmethylene)bis(3-methyl-1-phenyl-1<i>H</i>-pyrazol-5-ol) by Olalla Barreiro-Costa, Cristina Quiroga Lozano, Erika Muñoz, Patricio Rojas-Silva, Andrea Medeiros, Marcelo A. Comini, Jorge Heredia-Moya
Published in Biomedicines (2022-08-01)Get full text
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Selenosugars targeting the infective stage of Trypanosoma brucei with high selectivity by Estefanía Dibello, Natalia Oddone, Jaime Franco, Tünde-Zita Illyés, Andrea Medeiros, Attila Kiss, Fanni Hőgye, Katalin E. Kövér, László Szilágyi, Marcelo A. Comini
Published in International Journal for Parasitology: Drugs and Drug Resistance (2024-04-01)Get full text
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The indole motif is essential for the antitrypanosomal activity of N5-substituted paullones. by Irina Ihnatenko, Marco J Müller, Oliver C F Orban, Jens C Lindhof, Diego Benítez, Cecilia Ortíz, Estefanía Dibello, Leonardo L Seidl, Marcelo A Comini, Conrad Kunick
Published in PLoS ONE (2023-01-01)Get full text
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Drug-like molecules with anti-trypanothione synthetase activity identified by high throughput screening by Diego Benítez, Jaime Franco, Florencia Sardi, Alejandro Leyva, Rosario Durán, Gahee Choi, Gyongseon Yang, Taehee Kim, Namyoul Kim, Jinyeong Heo, Kideok Kim, Honggun Lee, Inhee Choi, Constantin Radu, David Shum, Joo Hwan No, Marcelo A. Comini
Published in Journal of Enzyme Inhibition and Medicinal Chemistry (2022-12-01)Get full text
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Identification of Novel Chemical Scaffolds Inhibiting Trypanothione Synthetase from Pathogenic Trypanosomatids. by Diego Benítez, Andrea Medeiros, Lucía Fiestas, Esteban A Panozzo-Zenere, Franziska Maiwald, Kyriakos C Prousis, Marina Roussaki, Theodora Calogeropoulou, Anastasia Detsi, Timo Jaeger, Jonas Šarlauskas, Lucíja Peterlin Mašič, Conrad Kunick, Guillermo R Labadie, Leopold Flohé, Marcelo A Comini
Published in PLoS Neglected Tropical Diseases (2016-04-01)Get full text
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Drug repurposing screening validated by experimental assays identifies two clinical drugs targeting SARS-CoV-2 main protease by Denis N. Prada Gori, Santiago Ruatta, Santiago Ruatta, Martín Fló, Martín Fló, Lucas N. Alberca, Carolina L. Bellera, Soonju Park, Jinyeong Heo, Honggun Lee, Kyu-Ho Paul Park, Otto Pritsch, Otto Pritsch, David Shum, Marcelo A. Comini, Alan Talevi
Published in Frontiers in Drug Discovery (2023-01-01)Get full text
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Garbage in, garbage out: how reliable training data improved a virtual screening approach against SARS-CoV-2 MPro by Santiago M. Ruatta, Santiago M. Ruatta, Denis N. Prada Gori, Martín Fló Díaz, Martín Fló Díaz, Franca Lorenzelli, Karen Perelmuter, Lucas N. Alberca, Lucas N. Alberca, Carolina L. Bellera, Carolina L. Bellera, Andrea Medeiros, Andrea Medeiros, Gloria V. López, Gloria V. López, Mariana Ingold, Williams Porcal, Williams Porcal, Estefanía Dibello, Irina Ihnatenko, Conrad Kunick, Marcelo Incerti, Martín Luzardo, Maximiliano Colobbio, Maximiliano Colobbio, Juan Carlos Ramos, Juan Carlos Ramos, Eduardo Manta, Eduardo Manta, Lucía Minini, María Laura Lavaggi, Paola Hernández, Jonas Šarlauskas, César Sebastian Huerta García, Rafael Castillo, Alicia Hernández-Campos, Giovanni Ribaudo, Giuseppe Zagotto, Renzo Carlucci, Noelia S. Medrán, Guillermo R. Labadie, Maitena Martinez-Amezaga, Carina M. L. Delpiccolo, Ernesto G. Mata, Laura Scarone, Laura Posada, Gloria Serra, Theodora Calogeropoulou, Kyriakos Prousis, Anastasia Detsi, Mauricio Cabrera, Guzmán Alvarez, Adrián Aicardo, Adrián Aicardo, Adrián Aicardo, Verena Araújo, Verena Araújo, Verena Araújo, Cecilia Chavarría, Cecilia Chavarría, Lucija Peterlin Mašič, Melisa E. Gantner, Melisa E. Gantner, Manuel A. Llanos, Manuel A. Llanos, Santiago Rodríguez, Luciana Gavernet, Luciana Gavernet, Soonju Park, Jinyeong Heo, Honggun Lee, Kyu-Ho Paul Park, Mariela Bollati-Fogolín, Otto Pritsch, Otto Pritsch, David Shum, Alan Talevi, Alan Talevi, Marcelo A. Comini
Published in Frontiers in Pharmacology (2023-06-01)Get full text
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