Search Results - Matthias Rottmann
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The Importance of Murine Models in Determining In Vivo Pharmacokinetics, Safety, and Efficacy in Antimalarial Drug Discovery by Glory Adebayo, Opeyemi I. Ayanda, Matthias Rottmann, Olusola S. Ajibaye, Gbolahan Oduselu, Julius Mulindwa, Olayinka O. Ajani, Oluwagbemiga Aina, Pascal Mäser, Ezekiel Adebiyi
Published in Pharmaceuticals (2025-03-01)Get full text
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Regioselective Synthesis of Potential Non-Quinonoid Prodrugs of Plasmodione: Antiparasitic Properties Against Two Hemoglobin-Feeding Parasites and Drug Metabolism Studies by Elena Cesar-Rodo, Baptiste Dupouy, Cécile Häberli, Jean-Marc Strub, David L. Williams, Pascal Mäser, Matthias Rottmann, Jennifer Keiser, Don Antoine Lanfranchi, Elisabeth Davioud-Charvet
Published in Molecules (2024-11-01)Get full text
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Genetic validation of PfFKBP35 as an antimalarial drug target by Basil T Thommen, Jerzy M Dziekan, Fiona Achcar, Seth Tjia, Armin Passecker, Katarzyna Buczak, Christin Gumpp, Alexander Schmidt, Matthias Rottmann, Christof Grüring, Matthias Marti, Zbynek Bozdech, Nicolas MB Brancucci
Published in eLife (2023-11-01)Get full text
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Translation of liver stage activity of M5717, a Plasmodium elongation factor 2 inhibitor: from bench to bedside by Akash Khandelwal, Francisca Arez, Paula M. Alves, Lassina Badolo, Catarina Brito, Christoph Fischli, Diana Fontinha, Claude Oeuvray, Miguel Prudêncio, Matthias Rottmann, Justin Wilkins, Özkan Yalkinoglu, Wilhelmina M. Bagchus, Thomas Spangenberg
Published in Malaria Journal (2022-05-01)Get full text
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Key Contributions by the Swiss Tropical and Public Health Institute Towards New and Better Drugs for Tropical Diseases by Pascal Mäser, Sonja Bernhard, Reto Brun, Christian Burri, Sébastien Gagneux, Manuel W. Hetzel, Marcel Kaiser, Christian Lengeler, Gerd Pluschke, Elisabeth Reus, Matthias Rottmann, Jürg Utzinger, Louisa Warryn, Sergio Wittlin, Jennifer Keiser
Published in CHIMIA (2023-09-01)Get full text
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Positive Charge in an Antimalarial Compound Unlocks Broad-Spectrum Antibacterial Activity by Maria Braun-Cornejo, Mitchell Platteschorre, Vincent de Vries, Patricia Bravo, Vidhisha Sonawane, Mostafa M. Hamed, Jörg Haupenthal, Norbert Reiling, Matthias Rottmann, Dennis Piet, Peter Maas, Eleonora Diamanti, Anna K. H. Hirsch
Published in JACS Au (2025-02-01)Get full text
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Targeting the Plasmodium falciparum IspE Enzyme by Eleonora Diamanti, Annina M. Steinbach, Lais P. de Carvalho, Henni-Karoliina Ropponen, Antoine Lacour, Rawia Hamid, Sidra Eisa, Patricia Bravo, Spyridon Bousis, Boris Illarionov, Markus Fischer, Mostafa M. Hamed, Nina C. Bach, Matthias Rottmann, Jana Held, Matthias Witschel, Stephan A. Sieber, Anna K. H. Hirsch
Published in ACS Omega (2024-10-01)Get full text
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An all-in-one pipeline for the in vitro discovery and in vivo testing of Plasmodium falciparum malaria transmission blocking drugs by Nicolas M. B. Brancucci, Christin Gumpp, Geert-Jan van Gemert, Xiao Yu, Armin Passecker, Flore Nardella, Basil T. Thommen, Marc Chambon, Gerardo Turcatti, Ludovic Halby, Benjamin Blasco, Maëlle Duffey, Paola B. Arimondo, Teun Bousema, Artur Scherf, Didier Leroy, Taco W. A. Kooij, Matthias Rottmann, Till S. Voss
Published in Nature Communications (2025-07-01)Get full text
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Polyamidoamine Nanoparticles for the Oral Administration of Antimalarial Drugs by Elisabet Martí Coma-Cros, Arnau Biosca, Joana Marques, Laura Carol, Patricia Urbán, Diana Berenguer, Maria Cristina Riera, Michael Delves, Robert E. Sinden, Juan José Valle-Delgado, Lefteris Spanos, Inga Siden-Kiamos, Paula Pérez, Krijn Paaijmans, Matthias Rottmann, Amedea Manfredi, Paolo Ferruti, Elisabetta Ranucci, Xavier Fernàndez-Busquets
Published in Pharmaceutics (2018-11-01)Get full text
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