Set-Up and Validation of a High Throughput Screening Method for Human Monoacylglycerol Lipase (MAGL) Based on a New Red Fluorescent Probe

Monoacylglycerol lipase (MAGL) is a serine hydrolase that has a key regulatory role in controlling the levels of 2-arachidonoylglycerol (2-AG), the main signaling molecule in the endocannabinoid system. Identification of selective modulators of MAGL enables both to provide new tools for investigatin...

書誌詳細
出版年:	Molecules
主要な著者:	Matteo Miceli, Silvana Casati, Roberta Ottria, Simone Di Leo, Ivano Eberini, Luca Palazzolo, Chiara Parravicini, Pierangela Ciuffreda
フォーマット:	論文
言語:	英語
出版事項:	MDPI AG 2019-06-01
主題:	high-throughput screening endocannabinoid monoacylglycerol lipase assay development
オンライン･アクセス:	https://www.mdpi.com/1420-3049/24/12/2241

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