Search Results - Adel S. El-Azab
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Synthesis and Conformational Analysis of Sterically Congested (4R)-(−)-1-(2,4,6-Trimethylbenzenesulfonyl)-3-n-butyryl-4-tert-butyl-2-imidazolidinone: X-Ray Crystallography and Semi... by Ibrahim A. Al-Swaidan, Adel S. El-Azab, Amer M. Alanazi, Alaa A.-M. Abdel-Aziz
Published in Journal of Chemistry (2014-01-01)Get full text
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An Alternative Route for Synthesis of Chiral 4-Substituted 1-Arenesulfonyl-2-imidazolidinones: Unusual Utility of (4S,5S)- and (4R,5R)-4,5-Dimethoxy-2-imidazolidinones and X-Ray Cr... by Ibrahim A. Al-Swaidan, Amer M. Alanazi, Adel S. El-Azab, Alaa A.-M. Abdel-Aziz
Published in Journal of Chemistry (2013-01-01)Get full text
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Synthesis of novel spirochromane incorporating Schiff's bases, potential antiproliferative activity, and dual EGFR/HER2 inhibition: Cell cycle analysis and in silico study by Dina I.A. Othman, Abdelrahman Hamdi, Walaa M. Elhusseiny, Adel S. El-Azab, Ahmed H. Bakheit, Mohamed Hefnawy, Alaa A.-M. Abdel-Aziz
Published in Saudi Pharmaceutical Journal (2023-11-01)Get full text
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Design, synthesis, and carbonic anhydrase inhibition activities of Schiff bases incorporating benzenesulfonamide scaffold: Molecular docking application by Adel S. El-Azab, Alaa A.-M. Abdel-Aziz, Silvia Bua, Alessio Nocentini, Ahmed H. Bakheit, Hamad M. Alkahtani, Mohamed M. Hefnawy, Claudiu T. Supuran
Published in Saudi Pharmaceutical Journal (2023-12-01)Get full text
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Synthesis, Antitumor Activities, and Apoptosis-Inducing Activities of Schiff’s Bases Incorporating Imidazolidine-2,4-dione Scaffold: Molecular Docking Studies and Enzymatic Inhibit... by Fhdah S. Alanazi, Hamad M. Alkahtani, Alaa A.-M. Abdel-Aziz, Adel S. El-Azab, Hanadi H. Asiri, Ahmed H. Bakheit, Fatmah A. Al-Omary
Published in Pharmaceuticals (2025-03-01)Get full text
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A Liquid Chromatography Tandem Mass Spectrometry Method for the Simultaneous Estimation of the Dopamine Receptor Antagonist LE300 and Its N-methyl Metabolite in Plasma: Application... by Mohamed M. Hefnawy, Mohamed W. Attwa, Adeeba A. Alzamil, Manal A. El-Gendy, Adel S. El-Azab, Yousef A. Bin Jardan, Ali A. El-Gamal
Published in Molecules (2023-02-01)Get full text
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Synthesis, anticancer and apoptosis-inducing activities of quinazoline–isatin conjugates: epidermal growth factor receptor-tyrosine kinase assay and molecular docking studies by Adel S. El-Azab, Abdullah Al-Dhfyan, Alaa A.-M. Abdel-Aziz, Laila A. Abou-Zeid, Hamad M. Alkahtani, Abdulrahman M. Al-Obaid, Manal A. Al-Gendy
Published in Journal of Enzyme Inhibition and Medicinal Chemistry (2017-01-01)Get full text
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A Rapid and Sensitive Liquid Chromatography-Tandem Mass Spectrometry Bioanalytical Method for the Quantification of Encorafenib and Binimetinib as a First-Line Treatment for Advanc... by Mohamed M. Hefnawy, Mohammed M. Alanazi, Abdullah M. Al-Hossaini, Abdulaziz I. Alnasser, Adel S. El-Azab, Yousef A. Bin Jardan, Mohamed W. Attwa, Manal A. El-Gendy
Published in Molecules (2022-12-01)Get full text
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Carbonic Anhydrase Inhibition Activities of Schiff’s Bases Based on Quinazoline-Linked Benzenesulfonamide by Adel S. El-Azab, Alaa A.-M. Abdel-Aziz, Hazem A. Ghabbour, Silvia Bua, Alessio Nocentini, Hamad M. Alkahtani, Nawaf A. Alsaif, Mohamed H. M. Al-Agamy, Claudiu T. Supuran
Published in Molecules (2022-11-01)Get full text
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Synthesis, Anticancer Screening of Some Novel Trimethoxy Quinazolines and VEGFR2, EGFR Tyrosine Kinase Inhibitors Assay; Molecular Docking Studies by Abdulmalik S. Altamimi, Adel S. El-Azab, Sami G. Abdelhamid, Mubarak A. Alamri, Ashraf H. Bayoumi, Safar M. Alqahtani, Alhumaidi B. Alabbas, Ali I. Altharawi, Manal A. Alossaimi, Menshawy A. Mohamed
Published in Molecules (2021-05-01)Get full text
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Synthesis, anticancer, apoptosis-inducing activities and EGFR and VEGFR2 assay mechanistic studies of 5,5-diphenylimidazolidine-2,4-dione derivatives: Molecular docking studies by Hamad M. Alkahtani, Mohammed M. Alanazi, Fadilah Sfouq Aleanizy, Fulwah Yahya Alqahtani, Ali Alhoshani, Fawaz E. Alanazi, Abdulrahman A. Almehizia, Ashraf N. Abdalla, Mashael G. Alanazi, Adel S. El-Azab, Alaa A.-M. Abdel-Aziz
Published in Saudi Pharmaceutical Journal (2019-07-01)Get full text
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LC–MS/MS method for the quantitation of decitabine and venetoclax in rat plasma after SPE: Application to pharmacokinetic study by Abdulaziz I. Alnasser, Mohamed M. Hefnawy, Abdullah M. Al-Hossaini, Yousef A. Bin Jardan, Adel S. El-Azab, Alaa M. Abdel-Aziz, Abdulrahman M. Al-Obaid, Ibrahim A. Al-Suwaidan, Mohamed W. Attwa, Manal A. El-Gendy
Published in Saudi Pharmaceutical Journal (2023-09-01)Get full text
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Synergistic Anti Leukemia Effect of a Novel Hsp90 and a Pan Cyclin Dependent Kinase Inhibitors by Ashraf N. Abdalla, Mohamed E. Abdallah, Akhmed Aslam, Ammar Bader, Antonio Vassallo, Nunziatina De Tommasi, Waleed H. Malki, Ahmed M. Gouda, Mohammed H. Mukhtar, Mahmoud Zaki El-Readi, Hamad M. Alkahtani, Alaa A.-M. Abdel-Aziz, Adel S. El-Azab
Published in Molecules (2020-05-01)Get full text
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Co-Inhibition of P-gp and Hsp90 by an Isatin-Derived Compound Contributes to the Increase of the Chemosensitivity of MCF7/ADR-Resistant Cells to Doxorubicin by Ashraf N. Abdalla, Miriana Di Stefano, Giulio Poli, Tiziano Tuccinardi, Ammar Bader, Antonio Vassallo, Mohamed E. Abdallah, Mahmoud Zaki El-Readi, Bassem Refaat, Alanood S. Algarni, Rizwan Ahmad, Hamad M. Alkahtani, Alaa A.-M. Abdel-Aziz, Adel S. El-Azab, Aljawharah Alqathama
Published in Molecules (2021-12-01)Get full text
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Synthesis, Cytotoxic Evaluation, and Structure-Activity Relationship of Substituted Quinazolinones as Cyclin-Dependent Kinase 9 Inhibitors by Hamad M. Alkahtani, Amer Alhaj Zen, Ahmad J. Obaidullah, Mohammed M. Alanazi, Abdulrahman A. Almehizia, Siddique Akber Ansari, Fadilah Sfouq Aleanizy, Fulwah Yahya Alqahtani, Rana M. Aldossari, Raghad Abdullah Algamdi, Lamees S. Al-Rasheed, Sami G. Abdel-Hamided, Alaa A.-M. Abdel-Aziz, Adel S. El-Azab
Published in Molecules (2022-12-01)Get full text
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