Search Results - Sandra Gemma
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Structure-Based Design of Biologically Active Compounds by Sandra Gemma
Published in Molecules (2020-07-01)Get full text
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Effects of structurally distinct human HDAC6 and HDAC6/HDAC8 inhibitors against S. mansoni larval and adult worm stages. by Roberto Gimmelli, Giuliana Papoff, Fulvio Saccoccia, Cristiana Lalli, Sandra Gemma, Giuseppe Campiani, Giovina Ruberti
Published in PLoS Neglected Tropical Diseases (2024-02-01)Get full text
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In Silico Analysis of Peptide-Based Derivatives Containing Bifunctional Warheads Engaging Prime and Non-Prime Subsites to Covalent Binding SARS-CoV-2 Main Protease (M<sup>pro</sup>... by Simone Brogi, Sara Rossi, Roberta Ibba, Stefania Butini, Vincenzo Calderone, Giuseppe Campiani, Sandra Gemma
Published in Computation (2022-05-01)Get full text
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Covalent Reversible Inhibitors of Cysteine Proteases Containing the Nitrile Warhead: Recent Advancement in the Field of Viral and Parasitic Diseases by Simone Brogi, Roberta Ibba, Sara Rossi, Stefania Butini, Vincenzo Calderone, Sandra Gemma, Giuseppe Campiani
Published in Molecules (2022-04-01)Get full text
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The green chemistry of chalcones: Valuable sources of privileged core structures for drug discovery by Ludovica Marotta, Sara Rossi, Roberta Ibba, Simone Brogi, Vincenzo Calderone, Stefania Butini, Giuseppe Campiani, Sandra Gemma
Published in Frontiers in Chemistry (2022-09-01)Get full text
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Unlocking the potential of biostimulants in sustainable agriculture: Effect of wood distillate on the nutritional profiling of apples by Riccardo Fedeli, Maria Dichiara, Gabriele Carullo, Valeria Tudino, Sandra Gemma, Stefania Butini, Giuseppe Campiani, Stefano Loppi
Published in Heliyon (2024-09-01)Get full text
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Development of Quinazolinone Derivatives as Modulators of Virulence Factors of <i>Pseudomonas aeruginosa</i> Cystic Fibrosis Strains by Gabriele Carullo, Giovanni Di Bonaventura, Sara Rossi, Veronica Lupetti, Valeria Tudino, Simone Brogi, Stefania Butini, Giuseppe Campiani, Sandra Gemma, Arianna Pompilio
Published in Molecules (2023-09-01)Get full text
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In Vitro and In Silico Analyses of New Cinnamid and Rosmarinic Acid-Derived Compounds Biosynthesized in <i>Escherichia coli</i> as <i>Leishmania amazonensis</i> Arginase Inhibitors by Julio Abel Alfredo dos Santos Simone Come, Yibin Zhuang, Tianzhen Li, Simone Brogi, Sandra Gemma, Tao Liu, Edson Roberto da Silva
Published in Pathogens (2022-09-01)Get full text
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Total Synthesis of the Natural Chalcone Lophirone E, Synthetic Studies toward Benzofuran and Indole-Based Analogues, and Investigation of Anti-Leishmanial Activity by Luca Pozzetti, Roberta Ibba, Sara Rossi, Orazio Taglialatela-Scafati, Donatella Taramelli, Nicoletta Basilico, Sarah D’Alessandro, Silvia Parapini, Stefania Butini, Giuseppe Campiani, Sandra Gemma
Published in Molecules (2022-01-01)Get full text
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Extra Virgin Olive Oil Extracts of Indigenous Southern Tuscany Cultivar Act as Anti-Inflammatory and Vasorelaxant Nutraceuticals by Luca Pozzetti, Francesca Ferrara, Ludovica Marotta, Sandra Gemma, Stefania Butini, Mascia Benedusi, Fabio Fusi, Amer Ahmed, Serena Pomponi, Stefano Ferrari, Matteo Perini, Anna Ramunno, Giacomo Pepe, Pietro Campiglia, Giuseppe Valacchi, Gabriele Carullo, Giuseppe Campiani
Published in Antioxidants (2022-02-01)Get full text
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Unveiling Wound Healing Properties of Biostimulated Walnut Kernel Extracts via Epithelial Mesenchymal Transition: Switching a Nutritional Matrix into a Therapeutic Remedy by Riccardo Fedeli, Elia Ranzato, Simona Martinotti, Manuela Giovanna Basilicata, Ludovica Marotta, Marianna Fava, Ilaria Cursaro, Giulio Tremori, Gregorio Bonsignore, Gabriele Carullo, Sandra Gemma, Giovanna Aquino, Pietro Campiglia, Giacomo Pepe, Stefania Butini, Stefano Loppi, Giuseppe Campiani
Published in Antioxidants (2025-09-01)Get full text
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Reversing TGF-β1-induced fibrotic phenotype in human lung fibroblasts using a PROTAC tool derived from an indoline-based HDAC6 inhibitor by Ilaria Cursaro, Valerio Ciccone, Valeria Tudino, Chiara Papulino, Laura Scalvini, Sandra Donnini, Lucia Morbidelli, Luca Bini, Claudia Landi, Chiara Contri, Silvia Pasquini, Fabrizio Vincenzi, Katia Varani, Alessio Lodola, Marco Mor, Rosaria Benedetti, Lucia Altucci, Stefania Butini, Gabriele Carullo, Sandra Gemma, Giuseppe Campiani
Published in European Journal of Medicinal Chemistry Reports (2025-08-01)Get full text
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