KUALA: a machine learning-driven framework for kinase inhibitors repositioning

Abstract The family of protein kinases comprises more than 500 genes involved in numerous functions. Hence, their physiological dysfunction has paved the way toward drug discovery for cancer, cardiovascular, and inflammatory diseases. As a matter of fact, Kinase binding sites high similarity has a d...

Full description

Bibliographic Details
Published in:Scientific Reports
Main Authors: Giada De Simone, Davide Stefano Sardina, Maria Rita Gulotta, Ugo Perricone
Format: Article
Language:English
Published: Nature Portfolio 2022-10-01
Online Access:https://doi.org/10.1038/s41598-022-22324-8