Molecular modelling and simulation studies of the Mycobacterium tuberculosis multidrug efflux pump protein Rv1258c.

Mycobacterial efflux pumps play a major role in the emergence of antimycobacterial drug resistance. Of particular interest is the proteinaceous multi-drug efflux pump protein Rv1258c that encodes a tetracycline/aminoglycoside resistance (TAP-2)-like efflux pump which is active in susceptible and dru...

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Bibliographic Details
Published in:PLoS ONE
Main Authors: Ruben Cloete, Erika Kapp, Jacques Joubert, Alan Christoffels, Sarel F Malan
Format: Article
Language:English
Published: Public Library of Science (PLoS) 2018-01-01
Online Access:https://doi.org/10.1371/journal.pone.0207605