Efficient Access to 3,5-Disubstituted 7-(Trifluoromethyl)pyrazolo[1,5-<i>a</i>]pyrimidines Involving S<i><sub>N</sub></i>Ar and Suzuki Cross-Coupling Reactions
An efficient and original synthesis of various 3,5-disubstituted 7-(trifluoromethyl)pyrazolo[1,5-<i>a</i>]pyrimidines is reported. A library of compounds diversely substituted in C-3 and C-5 positions was easily prepared from a common starting material, 3-bromo-7-(trifluoromethyl)pyrazol...
Main Authors: | Badr Jismy, Abdellatif Tikad, Mohamed Akssira, Gérald Guillaumet, Mohamed Abarbri |
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Format: | Article |
Language: | English |
Published: |
MDPI AG
2020-04-01
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Series: | Molecules |
Subjects: | |
Online Access: | https://www.mdpi.com/1420-3049/25/9/2062 |
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