Open Source Drug Discovery: Highly Potent Antimalarial Compounds Derived from the Tres Cantos Arylpyrroles
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| Format: | Article |
| Language: | English |
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American Chemical Society
2016-09-01
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| Series: | ACS Central Science |
| Online Access: | http://dx.doi.org/10.1021/acscentsci.6b00086 |
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DOAJ |
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English |
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Article |
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DOAJ |
| author |
Alice E. Williamson Paul M. Ylioja Murray N. Robertson Yevgeniya Antonova-Koch Vicky Avery Jonathan B. Baell Harikrishna Batchu Sanjay Batra Jeremy N. Burrows Soumya Bhattacharyya Felix Calderon Susan A. Charman Julie Clark Benigno Crespo Matin Dean Stefan L. Debbert Michael Delves Adelaide S. M. Dennis Frederik Deroose Sandra Duffy Sabine Fletcher Guri Giaever Irene Hallyburton Francisco-Javier Gamo Marinella Gebbia R. Kiplin Guy Zoe Hungerford Kiaran Kirk Maria J. Lafuente-Monasterio Anna Lee Stephan Meister Corey Nislow John P. Overington George Papadatos Luc Patiny James Pham Stuart A. Ralph Andrea Ruecker Eileen Ryan Christopher Southan Kumkum Srivastava Chris Swain Matthew J. Tarnowski Patrick Thomson Peter Turner Iain M. Wallace Timothy N. C. Wells Karen White Laura White Paul Willis Elizabeth A. Winzeler Sergio Wittlin Matthew H. Todd |
| spellingShingle |
Alice E. Williamson Paul M. Ylioja Murray N. Robertson Yevgeniya Antonova-Koch Vicky Avery Jonathan B. Baell Harikrishna Batchu Sanjay Batra Jeremy N. Burrows Soumya Bhattacharyya Felix Calderon Susan A. Charman Julie Clark Benigno Crespo Matin Dean Stefan L. Debbert Michael Delves Adelaide S. M. Dennis Frederik Deroose Sandra Duffy Sabine Fletcher Guri Giaever Irene Hallyburton Francisco-Javier Gamo Marinella Gebbia R. Kiplin Guy Zoe Hungerford Kiaran Kirk Maria J. Lafuente-Monasterio Anna Lee Stephan Meister Corey Nislow John P. Overington George Papadatos Luc Patiny James Pham Stuart A. Ralph Andrea Ruecker Eileen Ryan Christopher Southan Kumkum Srivastava Chris Swain Matthew J. Tarnowski Patrick Thomson Peter Turner Iain M. Wallace Timothy N. C. Wells Karen White Laura White Paul Willis Elizabeth A. Winzeler Sergio Wittlin Matthew H. Todd Open Source Drug Discovery: Highly Potent Antimalarial Compounds Derived from the Tres Cantos Arylpyrroles ACS Central Science |
| author_facet |
Alice E. Williamson Paul M. Ylioja Murray N. Robertson Yevgeniya Antonova-Koch Vicky Avery Jonathan B. Baell Harikrishna Batchu Sanjay Batra Jeremy N. Burrows Soumya Bhattacharyya Felix Calderon Susan A. Charman Julie Clark Benigno Crespo Matin Dean Stefan L. Debbert Michael Delves Adelaide S. M. Dennis Frederik Deroose Sandra Duffy Sabine Fletcher Guri Giaever Irene Hallyburton Francisco-Javier Gamo Marinella Gebbia R. Kiplin Guy Zoe Hungerford Kiaran Kirk Maria J. Lafuente-Monasterio Anna Lee Stephan Meister Corey Nislow John P. Overington George Papadatos Luc Patiny James Pham Stuart A. Ralph Andrea Ruecker Eileen Ryan Christopher Southan Kumkum Srivastava Chris Swain Matthew J. Tarnowski Patrick Thomson Peter Turner Iain M. Wallace Timothy N. C. Wells Karen White Laura White Paul Willis Elizabeth A. Winzeler Sergio Wittlin Matthew H. Todd |
| author_sort |
Alice E. Williamson |
| title |
Open Source Drug Discovery: Highly Potent Antimalarial Compounds Derived from the Tres Cantos Arylpyrroles |
| title_short |
Open Source Drug Discovery: Highly Potent Antimalarial Compounds Derived from the Tres Cantos Arylpyrroles |
| title_full |
Open Source Drug Discovery: Highly Potent Antimalarial Compounds Derived from the Tres Cantos Arylpyrroles |
| title_fullStr |
Open Source Drug Discovery: Highly Potent Antimalarial Compounds Derived from the Tres Cantos Arylpyrroles |
| title_full_unstemmed |
Open Source Drug Discovery: Highly Potent Antimalarial Compounds Derived from the Tres Cantos Arylpyrroles |
| title_sort |
open source drug discovery: highly potent antimalarial compounds derived from the tres cantos arylpyrroles |
| publisher |
American Chemical Society |
| series |
ACS Central Science |
| issn |
2374-7943 2374-7951 |
| publishDate |
2016-09-01 |
| url |
http://dx.doi.org/10.1021/acscentsci.6b00086 |
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doaj-389f0d71ee2a4fb79f8bb1da8028bfae2020-11-25T03:16:53ZengAmerican Chemical SocietyACS Central Science2374-79432374-79512016-09-0121068770110.1021/acscentsci.6b00086Open Source Drug Discovery: Highly Potent Antimalarial Compounds Derived from the Tres Cantos ArylpyrrolesAlice E. Williamson0Paul M. Ylioja1Murray N. Robertson2Yevgeniya Antonova-Koch3Vicky Avery4Jonathan B. Baell5Harikrishna Batchu6Sanjay Batra7Jeremy N. Burrows8Soumya Bhattacharyya9Felix Calderon10Susan A. Charman11Julie Clark12Benigno Crespo13Matin Dean14Stefan L. Debbert15Michael Delves16Adelaide S. M. Dennis17Frederik Deroose18Sandra Duffy19Sabine Fletcher20Guri Giaever21Irene Hallyburton22Francisco-Javier Gamo23Marinella Gebbia24R. Kiplin Guy25Zoe Hungerford26Kiaran Kirk27Maria J. Lafuente-Monasterio28Anna Lee29Stephan Meister30Corey Nislow31John P. Overington32George Papadatos33Luc Patiny34James Pham35Stuart A. Ralph36Andrea Ruecker37Eileen Ryan38Christopher Southan39Kumkum Srivastava40Chris Swain41Matthew J. Tarnowski42Patrick Thomson43Peter Turner44Iain M. Wallace45Timothy N. C. Wells46Karen White47Laura White48Paul Willis49Elizabeth A. Winzeler50Sergio Wittlin51Matthew H. Todd52School of Chemistry, The University of Sydney, Sydney, New South Wales, AustraliaSchool of Chemistry, The University of Sydney, Sydney, New South Wales, AustraliaSchool of Chemistry, The University of Sydney, Sydney, New South Wales, AustraliaDepartment of Pediatrics, Pharmacology & Drug Development, University of California San Diego, La Jolla, California, United StatesDiscovery Biology, Eskitis Institute for Drug Discovery, Griffith University, Nathan, Queensland, AustraliaMonash Institute of Pharmaceutical Sciences, Monash University, Parkville, Victoria, AustraliaCSIR-Central Drug Research Institute, Lucknow, IndiaCSIR-Central Drug Research Institute, Lucknow, IndiaMedicines for Malaria Venture, Geneva 15, SwitzerlandCSIR-Central Drug Research Institute, Lucknow, IndiaTres Cantos Medicines Development Campus, Diseases of the Developing World, GlaxoSmithKline, Tres Cantos, SpainMonash Institute of Pharmaceutical Sciences, Monash University, Parkville, Victoria, AustraliaDepartment of Chemical Biology & Therapeutics, St. Jude Children’s Research Hospital, Memphis, Tennessee, United StatesTres Cantos Medicines Development Campus, Diseases of the Developing World, GlaxoSmithKline, Tres Cantos, SpainSchool of Chemistry, The University of Sydney, Sydney, New South Wales, AustraliaDepartment of Chemistry, Lawrence University, Appleton, Wisconsin, United StatesDepartment of Life Sciences, Imperial College London, London, U.K.Research School of Biology, The Australian National University, Canberra, AustraliaAsclepia Outsourcing Solutions, Destelbergen, BelgiumDiscovery Biology, Eskitis Institute for Drug Discovery, Griffith University, Nathan, Queensland, AustraliaDiscovery Biology, Eskitis Institute for Drug Discovery, Griffith University, Nathan, Queensland, AustraliaDonnelly Centre for Cellular and Biomolecular Research, University of Toronto, Toronto, Ontario, CanadaDrug Discovery Unit, Division of Biological Chemistry and Drug Discovery, University of Dundee, Dundee, U.K.Tres Cantos Medicines Development Campus, Diseases of the Developing World, GlaxoSmithKline, Tres Cantos, SpainDonnelly Centre for Cellular and Biomolecular Research, University of Toronto, Toronto, Ontario, CanadaDepartment of Chemical Biology & Therapeutics, St. Jude Children’s Research Hospital, Memphis, Tennessee, United StatesSchool of Chemistry, The University of Sydney, Sydney, New South Wales, AustraliaResearch School of Biology, The Australian National University, Canberra, AustraliaTres Cantos Medicines Development Campus, Diseases of the Developing World, GlaxoSmithKline, Tres Cantos, SpainDonnelly Centre for Cellular and Biomolecular Research, University of Toronto, Toronto, Ontario, CanadaDepartment of Pediatrics, Pharmacology & Drug Development, University of California San Diego, La Jolla, California, United StatesDonnelly Centre for Cellular and Biomolecular Research, University of Toronto, Toronto, Ontario, CanadaEuropean Molecular Biology LaboratoryEuropean Bioinformatics Institute, Hinxton, Cambridgeshire, U.K.European Molecular Biology LaboratoryEuropean Bioinformatics Institute, Hinxton, Cambridgeshire, U.K.Institute of Chemical Sciences and Engineering (ISIC), Ecole Polytechnique Fédérale de Lausanne (EPFL), Lausanne, SwitzerlandDepartment of Biochemistry & Molecular Biology, Bio21 Molecular Science and Biotechnology Institute, The University of Melbourne, Melbourne, Victoria, AustraliaDepartment of Biochemistry & Molecular Biology, Bio21 Molecular Science and Biotechnology Institute, The University of Melbourne, Melbourne, Victoria, AustraliaDepartment of Life Sciences, Imperial College London, London, U.K.Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, Victoria, AustraliaIUPHAR/BPS Guide to PHARMACOLOGY, Centre for Integrative Physiology, School of Biomedical Sciences, University of Edinburgh, Edinburgh, U.K.CSIR-Central Drug Research Institute, Lucknow, IndiaCambridge MedChem Consulting, Duxford, Cambridge, U.K.School of Chemistry, The University of Sydney, Sydney, New South Wales, AustraliaSchool of Chemistry, The University of Edinburgh, Edinburgh, U.K.School of Chemistry, The University of Sydney, Sydney, New South Wales, AustraliaEuropean Molecular Biology LaboratoryEuropean Bioinformatics Institute, Hinxton, Cambridgeshire, U.K.Medicines for Malaria Venture, Geneva 15, SwitzerlandMonash Institute of Pharmaceutical Sciences, Monash University, Parkville, Victoria, AustraliaSchool of Chemistry, The University of Sydney, Sydney, New South Wales, AustraliaMedicines for Malaria Venture, Geneva 15, SwitzerlandDepartment of Pediatrics, Pharmacology & Drug Development, University of California San Diego, La Jolla, California, United StatesSwiss Tropical and Public Health Institute, Basel, SwitzerlandSchool of Chemistry, The University of Sydney, Sydney, New South Wales, Australiahttp://dx.doi.org/10.1021/acscentsci.6b00086 |