Synthesis and Fungicidal Activity of Novel 2,3-Disubstituted-1,3-benzoxazines

Synthesis and Fungicidal Activity of Novel 2,3-Disubstituted-1,3-benzoxazines

A series of new 2,3-disubstituted-3,4-dihydro-2<em>H</em>-1,3-benzoxazines were prepared in moderate to excellent yields by aza-acetalizations of aromatic aldehydes with 2-(<em>N</em>-substituted aminomethyl)phenols in the presence of TMSCl. Th...

Full description

Bibliographic Details
Main Authors:	Xiaoming Ou, Jinwen Chen, Wenjing Xiao, Hanwen Liu, Zanwen Xia, Zhonghua Zhu, Zilong Tang
Format:	Article
Language:	English
Published:	MDPI AG 2012-07-01
Series:	Molecules
Subjects:	2,3-disubstituted-1,3-benzoxazine synthesis chlorotrimethylsilane fungicidal activity
Online Access:	http://www.mdpi.com/1420-3049/17/7/8174

Similar Items

Synthesis and Fungicidal Activity of 1-(Carbamoylmethyl)-2-aryl-3,1-benzoxazines
by: Zi-Long Tang, et al.
Published: (2017-07-01)

3,4-Dihydro-2H-1,3-benzoxazines and their oxo-derivatives - Chemistry and bioactivities
by: Sharaf El-Din Nabaweya Abd El-Salam
Published: (2021-01-01)

Developing Further Versatility in Benzoxazine Synthesis via Hydrolytic Ring-Opening
by: Shaoying Cui, et al.
Published: (2020-03-01)

Direct Synthesis of Phosphonates and α-Amino-phosphonates from 1,3-Benzoxazines
by: Oscar Salgado-Escobar, et al.
Published: (2019-01-01)

Diethyl 3-amino-6-methyl-4-[(E)-2-phenylethenyl]thieno[2,3-b]pyridine-2,5-dicarboxylate
by: Joel T. Mague, et al.
Published: (2016-02-01)

Synthesis of single stereoisomers of 2,2-disubstituted 3-hydroxycyclohexane-1-ones via enzymatic desymmetric reduction of the 1,3-cyclohexanediones
by: Liangyan Zhu, et al.
Published: (2021-08-01)

Synthesis of some Heterocyclic Compounds from 1,4-Benzoxazine-3-one
by: Omar A. Salih
Published: (2013-03-01)

Benzoxazine Monomers and Polymers Based on 3,3′-Dichloro-4,4′-Diaminodiphenylmethane: Synthesis and Characterization
by: Viktoria V. Petrakova, et al.
Published: (2021-04-01)

Synthesis and antimicrobial evaluation of 1,4-disubstituted 1,2,3-triazoles with aromatic ester functionality
by: C.P. Kaushik, et al.
Published: (2016-11-01)

Ascorbic Acid-Initiated Tandem Radical Cyclization of N-Arylacrylamides to Give 3,3-Disubstituted Oxindoles
by: Sheng Liu, et al.
Published: (2015-08-01)

Simple grinding-induced reactions of 2-aminobenzyl alcohol and benzaldehyde derivatives, a rapid synthetic route to 3,1-benzoxazines
by: I. B. Masesane, et al.
Published: (2014-05-01)

Synthesis of Chiral 1,4-Disubstituted-1,2,3-Triazole Derivatives from Amino Acids
by: Morten Grøtli, et al.
Published: (2009-12-01)

Crystal structure and C—H...F hydrogen bonding in the fluorinated bis-benzoxazine: 3,3′-(ethane-1,2-diyl)bis(6-fluoro-3,4-dihydro-2H-1,3-benzoxazine)
by: Augusto Rivera, et al.
Published: (2016-10-01)

Novel epoxy-benzoxazine water-based emulsions with reactive benzoxazine surfactants for coatings
by: M. Krajnc, et al.
Published: (2014-08-01)

3,1-Benzothiazines, 1,4-Benzodioxines and 1,4-Benzoxazines as Inhibitors of Matriptase-2: Outcome of a Focused Screening Approach
by: Polya G. Roydeva, et al.
Published: (2016-01-01)

Crystal structure of 3-(4-hydroxyphenyl)-2-[(E)-2-phenylethenyl]quinazolin-4(3H)-one
by: Inese Mierina, et al.
Published: (2016-04-01)

Various Synthetic Pathways for the Synthesis of 3,4-Disubstituted Isoxazole by One Pot Multicomponent Reaction
by: Parul Setia, et al.
Published: (2020-12-01)

Design, synthesis and biological evaluation of tricyclic pyrazolo[1,5-c][1,3]benzoxazin-5(5H)-one scaffolds as selective BuChE inhibitors
by: Guo-Liang Qiu, et al.
Published: (2018-01-01)

Design and Effects of the Cinnamic Acids Chemical Structures as Organocatalyst on the Polymerization of Benzoxazines
by: Rocío B. Rodríguez, et al.
Published: (2020-07-01)

Crystallographic and Spectroscopic Investigations on Oxidative Coordination in the Heteroleptic Mononuclear Complex of Cerium and Benzoxazine Dimer
by: Worawat Wattanathana, et al.
Published: (2021-09-01)

Benzoxazine Copolymers with Mono- and Difunctional Epoxy Active Diluents with Enhanced Tackiness and Reduced Viscosity
by: Natalia V. Bornosuz, et al.
Published: (2021-09-01)

Regioselective synthesis, characterization and antimicrobial evaluation of amide-ether linked 1,4-disubstituted 1,2,3-triazoles
by: Kaushik Chander Prakash, et al.
Published: (2017-01-01)

Design, Synthesis and Biological Evaluation of 1,4-Disubstituted-3,4-dihydroisoquinoline Compounds as New Tubulin Polymerization Inhibitors
by: Ling Zhang, et al.
Published: (2015-05-01)

Hepatotoxicity and antioxidant activity of some new N,N′-disubstituted benzimidazole-2-thiones, radical scavenging mechanism and structure-activity relationship
by: Neda O. Anastassova, et al.
Published: (2018-03-01)

A facile synthesis and fungicidal activities of 2-(alkylamino)-5,6-dimethylthieno[2,3-d]pyrimidin-4(3H)-ones
by: Yang-Gen Hu, et al.
Published: (2008-12-01)

Copolymers of Vinyl-Containing Benzoxazine with Vinyl Monomers as Precursors for High Performance Thermosets
by: Tsutomu Takeichi, et al.
Published: (2015-04-01)

Main Chain Type Benzoxazine Polymers for High Performance Applications
by: Chernykh, Andrey
Published: (2009)

Microwave Irradiation Promoted Reactions of Benzoxazin-4-Ones with Primary Amines. Preparation of 4(2=3H)-Quinazolinones
by: Mohammad Sadegh Khajavi, et al.
Published: (1999-06-01)

Recent Progress of High Performance Thermosets Based on Norbornene Functional Benzoxazine Resins
by: Yin Lu, et al.
Published: (2021-04-01)

Study on an amine-containing benzoxazine: Homo- and copolymerization with epoxy resin
by: L. Zhang, et al.
Published: (2016-07-01)

Synthesis of Novel Benzoxazines Containing Sulfur and Their Application in Rubber Compounds
by: Acerina Trejo-Machin, et al.
Published: (2021-04-01)

Produção conjunta de 1,3-Propanodiol e 2,3-Butanodiol por Klebsiella pneumoniae a partir de glicerina residual proveniente da fabricação de biodiesel
by: Rogério da Silva Santos
Published: (2013)

Produção conjunta de 1,3-Propanodiol e 2,3-Butanodiol por Klebsiella pneumoniae a partir de glicerina residual proveniente da fabricação de biodiesel
by: Santos, Rogério da Silva
Published: (2013)

Synthesis of Eugenol-Based Silicon-Containing Benzoxazines and Their Applications as Bio-Based Organic Coatings
by: Jinyue Dai, et al.
Published: (2018-02-01)

Review on the Accelerated and Low-Temperature Polymerization of Benzoxazine Resins: Addition Polymerizable Sustainable Polymers
by: Bimlesh Lochab, et al.
Published: (2021-04-01)

Silica-bound benzoyl chloride mediated the solid-phase synthesis of 4H-3,1-benzoxazin-4-ones
by: Kurosh Rad-Moghadam, et al.
Published: (2009-04-01)

Ring-Opening Polymerization of 1,3-Benzoxazines via Borane Catalyst
by: Mustafa Arslan, et al.
Published: (2018-02-01)

Microwave Assisted Synthesis of 2,2'-Arylene-substituted Bis(4H-3,1-Benzoxazin-4-one) Derivatives Using the Complex Cyanuric Chloride/N,N-Dimethylformamide
by: Mehdi Shariat, et al.
Published: (2012-09-01)

Multifunctional Benzoxazines Feature Low Polymerization Temperature and Diverse Polymer Structures
by: Marc Soto, et al.
Published: (2016-08-01)

Identification of Fungicidal 2,6-Disubstituted Quinolines with Activity against Candida Biofilms
by: Bruno P. A. Cammue, et al.
Published: (2012-10-01)