Pharmacological Profile of the Novel Anti-inflammatory Corticosteroid NS-126, a Therapeutic Agent for Allergic Rhinitis

NS-126 (9-fluoro-11β,17,21-trihydroxy-16α-methylpregna-1,4-diene-3,20-dione 21-cyclohexanecarboxylate 17-cyclopropanecarboxylate) is a novel, highly lipophilic anti-inflammatory corticosteroid. We compared NS-126 and the widely used intranasal corticosteroid fluticasone propionate (FP) in a guinea-p...

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Main Authors: Naoki Inoue, Asami Hashino, Kiyoto Kageyama, Xin Zhang, Takahiro Sasagawa, Naoko Kawakita, Yosuke Takahashi, Katsumi Yoshida, Mikiko Hashimoto, Kazuya Mori, Takashi Kyoi
Format: Article
Language:English
Published: Elsevier 2010-01-01
Series:Journal of Pharmacological Sciences
Online Access:http://www.sciencedirect.com/science/article/pii/S134786131931059X