Ethyl 2-[2-(4-Nitrobenzoyl)-1H-indol-3-yl]acetate

Ethyl 2-[2-(4-Nitrobenzoyl)-1H-indol-3-yl]acetate

Ethyl 2-[2-(4-nitrobenzoyl)-1H-indol-3-yl]acetate was prepared in good yield and characterized by the aza-alkylation/intramolecular Michael cascade reaction of (E)-ethyl 3-[2-(tosylamino)phenyl]acrylate with 2-bromo-4′′-nitroacetophenone, followed by desulfonative dehydrogenation with 1,8-diazabicyc...

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Bibliographic Details
Main Authors:	Sunyoung Choi, Sung-Gon Kim
Format:	Article
Language:	English
Published:	MDPI AG 2017-07-01
Series:	Molbank
Subjects:	Indole Michael reaction dehydrogenation cascade reaction
Online Access:	https://www.mdpi.com/1422-8599/2017/3/M945

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