Design, Synthesis, and Biological Evaluation of Novel Thienopyrimidine Derivatives as PI3Kα Inhibitors

Three series of novel thienopyrimidine derivatives <b>9a</b>&#8722;<b>l</b>, <b>15a</b>&#8722;<b>l</b>, and <b>18a</b>&#8722;<b>h</b> were designed and synthesized, and their IC<sub>50</sub> values agains...

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Bibliographic Details
Main Authors: Lide Yu, Qinqin Wang, Caolin Wang, Binliang Zhang, Zunhua Yang, Yuanying Fang, Wufu Zhu, Pengwu Zheng
Format: Article
Language:English
Published: MDPI AG 2019-09-01
Series:Molecules
Subjects:
Online Access:https://www.mdpi.com/1420-3049/24/19/3422