TDAE Strategy for the Synthesis of 2,3-Diaryl N-Tosylaziridines

We report herein an original and rapid synthesis of 2,3-diaryl N-tosylaziridines by TDAE strategy starting from ortho- or para-nitro(dichloromethyl)benzene derivatives and N-tosylimines. A mixture of cis/trans isomers was isolated from 1-(dichloromethyl)-4-nitrobenzene, whereas only trans-aziridines...

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Bibliographic Details
Main Authors: Thierry Terme, Cédric Spitz, Omar Khoumeri, Patrice Vanelle
Format: Article
Language:English
Published: MDPI AG 2013-06-01
Series:Molecules
Subjects:
Online Access:http://www.mdpi.com/1420-3049/18/7/7364