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01568 am a22002653u 4500 |
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72118 |
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|a dc
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|a Henderson, Jaclyn L.
|e author
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|a Massachusetts Institute of Technology. Department of Chemistry
|e contributor
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|a Massachusetts Institute of Technology. Department of Humanities. History Section
|e contributor
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|a Buchwald, Stephen L.
|e contributor
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|a Henderson, Jaclyn L.
|e contributor
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|a McDermott, Sarah M.
|e contributor
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|a Buchwald, Stephen Leffler
|e contributor
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|a McDermott, Sarah M.
|e author
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|a Buchwald, Stephen Leffler
|e author
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|a Palladium-Catalyzed Amination of Unprotected Halo-7- azaindoles
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|b American Chemical Society (ACS),
|c 2012-08-14T16:04:11Z.
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|z Get fulltext
|u http://hdl.handle.net/1721.1/72118
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|a Simple and efficient procedures for the Pd-catalyzed cross-coupling of primary and secondary amines with halo-7-azaindoles(pyrrolo[2,3-b]pyridine) are presented. Previously, no general method was available to ensure the highly selective reaction of the heteroaryl halide in the presence of the unprotected azaindole N-H. Using palladium precatalysts recently reported by our group, such reactions are easily accomplished under mild conditions that can be applied to cross-coupling reactions with a wide array of aliphatic and aromatic amines.
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|a Amgen, Inc.
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|a National Institutes of Health (U.S.) (Grant number GM-58160)
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|a en_US
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|a Article
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| 773 |
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|t Organic Letters
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