Palladium-Catalyzed Amination of Unprotected Halo-7- azaindoles
Simple and efficient procedures for the Pd-catalyzed cross-coupling of primary and secondary amines with halo-7-azaindoles(pyrrolo[2,3-b]pyridine) are presented. Previously, no general method was available to ensure the highly selective reaction of the heteroaryl halide in the presence of the unprot...
Main Authors: | Henderson, Jaclyn L. (Contributor), McDermott, Sarah M. (Contributor), Buchwald, Stephen Leffler (Contributor) |
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Other Authors: | Massachusetts Institute of Technology. Department of Chemistry (Contributor), Massachusetts Institute of Technology. Department of Humanities. History Section (Contributor), Buchwald, Stephen L. (Contributor) |
Format: | Article |
Language: | English |
Published: |
American Chemical Society (ACS),
2012-08-14T16:04:11Z.
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Subjects: | |
Online Access: | Get fulltext |
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