Design, synthesis and biological evaluation of TG2 transglutaminase inhibitors
La transglutaminase tissulaire (TG2) est une enzyme de la famille des transglutaminases (EC 2.3.2.13) qui est exprimée de manière ubiquitaire chez les mammifères. Cette enzyme catalyse la formation d'une liaison amide intra- ou intermoléculaire entre un résidu glutamine et un résidu lysine. Ce...
Main Author: | Fidalgo Lopez, Javier |
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Other Authors: | Lyon |
Language: | en |
Published: |
2016
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Subjects: | |
Online Access: | http://www.theses.fr/2016LYSE1190/document |
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