A class of carbonic anhydrase IX/XII – selective carboxylate inhibitors

by Rakia Abd Alhameed, Emanuela Berrino, Zainab Almarhoon, Ayman El-Faham, Claudiu T. Supuran
Published 2020-01-01

The antibiotic furagin and its derivatives are isoform-selective human carbonic anhydrase inhibitors

by Aleksandrs Pustenko, Alessio Nocentini, Paola Gratteri, Alessandro Bonardi, Igor Vozny, Raivis Žalubovskis, Claudiu T. Supuran
Published 2020-01-01

Aryl derivatives of 3H-1,2-benzoxathiepine 2,2-dioxide as carbonic anhydrase inhibitors

by Aleksandrs Pustenko, Alessio Nocentini, Anastasija Balašova, Ahmed Alafeefy, Mikhail Krasavin, Raivis Žalubovskis, Claudiu T. Supuran
Published 2020-01-01

7-Acylamino-3H-1,2-benzoxathiepine 2,2-dioxides as new isoform-selective carbonic anhydrase IX and XII inhibitors

by Aleksandrs Pustenko, Alessio Nocentini, Anastasija Balašova, Mikhail Krasavin, Raivis Žalubovskis, Claudiu T. Supuran
Published 2020-01-01

Benzamide-4-Sulfonamides Are Effective Human Carbonic Anhydrase I, II, VII, and IX Inhibitors

by Morteza Abdoli, Murat Bozdag, Andrea Angeli, Claudiu T. Supuran
Published 2018-06-01

Sulfocoumarins as dual inhibitors of human carbonic anhydrase isoforms IX/XII and of human thioredoxin reductase

by Mikhail Krasavin, Raivis Žalubovskis, Aiga Grandāne, Ilona Domračeva, Petr Zhmurov, Claudiu T. Supuran
Published 2020-01-01

Potent and Selective Carboxylic Acid Inhibitors of Tumor-Associated Carbonic Anhydrases IX and XII

by Ylenia Cau, Daniela Vullo, Mattia Mori, Elena Dreassi, Claudiu T. Supuran, Maurizio Botta
Published 2017-12-01

Extending the Inhibition Profiles of Coumarin-Based Compounds Against Human Carbonic Anhydrases: Synthesis, Biological, and In Silico Evaluation

by Victor Kartsev, Athina Geronikaki, Silvia Bua, Alessio Nocentini, Anthi Petrou, Boris Lichitsky, Mykhaylo Frasinyuk, Janis Leitans, Andris Kazaks, Kaspars Tars, Claudiu T. Supuran
Published 2019-10-01

Activation of carbonic anhydrase isoforms involved in modulation of emotional memory and cognitive...

by Gustavo Provensi, Alessio Nocentini, Maria Beatrice Passani, Patrizio Blandina, Claudiu T. Supuran
Published 2021-01-01

Organoruthenium(II) complexes of acetazolamide potently inhibit human carbonic anhydrase isoforms I, II, IX and XII

by Sara Seršen, Katja Traven, Jakob Kljun, Iztok Turel, Claudiu T. Supuran
Published 2019-01-01

3D QSAR studies, pharmacophore modeling, and virtual screening of diarylpyrazole–benzenesulfonamide derivatives as a template to obtain new inhibitors, using human carbonic anhydra...

by Yeganeh Entezari Heravi, Hassan Sereshti, Ali Akbar Saboury, Jahan Ghasemi, Marzieh Amirmostofian, Claudiu T. Supuran
Published 2017-01-01

Plasmatic carbonic anhydrase IX as a diagnostic marker for clear cell renal cell carcinoma

by Laura Lucarini, Lucia Magnelli, Nicola Schiavone, Alfonso Crisci, Alessio Innocenti, Luca Puccetti, Fabio Cianchi, Sara Peri, Claudiu T. Supuran, Laura Papucci, Emanuela Masini
Published 2018-01-01

Open saccharin-based secondary sulfonamides as potent and selective inhibitors of cancer-related carbonic anhydrase IX and XII isoforms

by Melissa D’Ascenzio, Paolo Guglielmi, Simone Carradori, Daniela Secci, Rosalba Florio, Adriano Mollica, Mariangela Ceruso, Atilla Akdemir, Anatoly P. Sobolev, Claudiu T. Supuran
Published 2017-01-01

Psychoactive substances belonging to the amphetamine class potently activate brain carbonic anhydrase isoforms VA, VB, VII, and XII

by Andrea Angeli, Fabio Vaiano, Francesco Mari, Elisabetta Bertol, Claudiu T. Supuran
Published 2017-01-01

Synthesis and biological evaluation of novel 3-(quinolin-4-ylamino)benzenesulfonamides as carbonic anhydrase isoforms I and II inhibitors

by Mohammad M. Al-Sanea, Ahmed Elkamhawy, Sora Paik, Silvia Bua, So Ha Lee, Mohamed A. Abdelgawad, Eun Joo Roh, Wagdy M. Eldehna, Claudiu T. Supuran
Published 2019-01-01

Primary mono- and bis-sulfonamides obtained via regiospecific sulfochlorination of N-arylpyrazoles: inhibition profile against a panel of human carbonic anhydrases

by Mikhail Krasavin, Mikhail Korsakov, Oksana Ronzhina, Tiziano Tuccinardi, Stanislav Kalinin, Muhammet Tanç, Claudiu T. Supuran
Published 2017-01-01

3H-1,2-benzoxathiepine 2,2-dioxides: a new class of isoform-selective carbonic anhydrase inhibitors

by Aleksandrs Pustenko, Dmitrijs Stepanovs, Raivis Žalubovskis, Daniela Vullo, Andris Kazaks, Janis Leitans, Kaspars Tars, Claudiu T. Supuran
Published 2017-01-01

Discovery of curcumin inspired sulfonamide derivatives as a new class of carbonic anhydrase isoforms I, II, IX, and XII inhibitors

by P. V. Sri Ramya, Srinivas Angapelly, Andrea Angeli, Chander Singh Digwal, Mohammed Arifuddin, Bathini Nagendra Babu, Claudiu T. Supuran, Ahmed Kamal
Published 2017-01-01

Activation of α-, β-, γ- δ-, ζ- and η- class of carbonic anhydrases with amines and amino acids: a review

by Suleyman Akocak, Claudiu T. Supuran
Published 2019-01-01

Indole-Based Hydrazones Containing A Sulfonamide Moiety as Selective Inhibitors of Tumor-Associated Human Carbonic Anhydrase Isoforms IX and XII

by Kübra Demir-Yazıcı, Silvia Bua, Nurgül Mutlu Akgüneş, Atilla Akdemir, Claudiu T. Supuran, Özlen Güzel-Akdemir
Published 2019-05-01