Mutations in pmrB Confer Cross-Resistance between the LptD Inhibitor POL7080 and Colistin in Pseudomonas aeruginosa

by Romano, Keith P., Warrier, Thulasi, Poulsen, Bradley E., Nguyen, Phuong H., Loftis, Alexander R., Saebi, Azin, Pentelute, Bradley L., Hung, Deborah T
Published 2020

Studies on a landscape of perfluoroaromatic-reactive peptides

by Evans, Ethan Daniel, Pentelute, Bradley L.
Published 2018

Total synthesis and biochemical characterization of mirror image barnase

by Vinogradov, Alexander Alexandrovich, Evans, Ethan Daniel, Pentelute, Bradley L.
Published 2017

Site-Selective Cysteine-Cyclooctyne Conjugation

by Zhang, Chi, Dai, Peng, Vinogradov, Alexander A., Gates, Zachary P, Pentelute, Bradley L.
Published 2020

Palladium Oxidative Addition Complexes for Peptide and Protein Cross-linking

by Kubota, Koji, Dai, Peng, Pentelute, Bradley L., Buchwald, Stephen Leffler
Published 2020

Efficient Flow Synthesis of Human Antimicrobial Peptides

by Albin, John S, Pentelute, Bradley L.
Published 2020

Synthesis of proteins by automated flow chemistry

by Hartrampf, Nina, Saebi, Azin, Poskus, M., Gates, Zachary P, Callahan, A. J., Cowfer, A. E., Hanna, S., Antilla, S., Schissel, Carly K., Quartararo, Anthony James, Ye, Xiyun, Mijalis, Alexander James, Simon, M. D., Loas, Andrei Ioan, Liu, S., Jessen, C., Nielsen, T. E., Pentelute, Bradley L.
Published 2020

Perfluoroaryl Bicyclic Cell-Penetrating Peptides for Delivery of Antisense Oligonucleotides

by Wolfe, Justin, Fadzen, Colin M., Holden, Rebecca Lynn, Yao, Monica, Hanson, Gunnar J., Pentelute, Bradley L.
Published 2020

Secondary Amino Alcohols: Traceless Cleavable Linkers for Use in Affinity Capture and Release

by Pomplun, Sebastian Johannes, Shugrue, Christopher R., Schmitt, Adeline M., Schissel, Carly K., Farquhar, Charlotte E., Pentelute, Bradley L.
Published 2020

Blood-brain-barrier spheroids as an in vitro screening platform for brain-penetrating agents

by Calligaris, David, Hornburg, Kalvis, Chiocca, E. Antonio, Agar, Nathalie Y. R., Lawler, Sean E., Cho, Choi-Fong, Wolfe, Justin, Fadzen, Colin M., Pentelute, Bradley L.
Published 2018

De Novo Discovery of High-Affinity Peptide Binders for the SARS-CoV-2 Spike Protein

by Pomplun, Sebastian Johannes, Jbara, Muhammad, Quartararo, Anthony James, Zhang, Genwei, Brown, Joseph S., Lee, Yen-Chun, Ye, Xiyun, Hanna, Stephanie, Pentelute, Bradley L.
Published 2021

A Perfluoroaryl-Cysteine S[subscript N]Ar Chemistry Approach to Unprotected Peptide Stapling

by Spokoyny, Alexander M., Zou, Yekui, Yu, Hongtao, Lin, Yu-Shan, Pentelute, Bradley L., Ling, Jingjing
Published 2015

Mucosal absorption of therapeutic peptides by harnessing the endogenous sorting of glycosphingolipids

by Garcia-Castillo, Maria Daniela, Chinnapen, Daniel J F, te Welscher, Yvonne M, Gonzalez, Rodrigo J, Softic, Samir, Pacheco, Michele, Mrsny, Randall J, Kahn, C Ronald, von Andrian, Ulrich H, Lau, Jesper, Pentelute, Bradley L., Lencer, Wayne I
Published 2020

A chemoselective strategy for late-stage functionalization of complex small molecules with polypeptides and proteins

by Cohen, Daniel Tzvi, Zhang, Chi, Fadzen, Colin M., Mijalis, Alexander James, Hie, Liana, Johnson, Kenneth D., Shriver, Zachary, Plante, Obadiah, Miller, Scott J., Buchwald, Stephen Leffler, Pentelute, Bradley L.
Published 2020

Conformational Stabilization and Rapid Labeling of a 29-Residue Peptide by a Small Molecule Reaction Partner

by Evans, Ethan Daniel, Gates, Zachary P, Sun, Zhen-Yu J., Mijalis, Alexander James, Pentelute, Bradley L.
Published 2020

Designing Well-Structured Cyclic Pentapeptides Based on Sequence-Structure Relationships

by Slough, Diana P., McHugh, Sean M., Cummings, Ashleigh E., Dal, Peng, Pentelute, Bradley L., Kritzer, Joshua A., Lin, Yu-Shan
Published 2020

Divergent unprotected peptide macrocyclisation by palladium-mediated cysteine arylation

by Reilly, John, Rojas, Anthony Jose, Zhang, Chi, Vinogradova, Ekaterina V., Buchwald, Nathan, Pentelute, Bradley L., Buchwald, Stephen Leffler
Published 2018

Blood-brain-barrier organoids for investigating the permeability of CNS therapeutics

by Bergmann, Sonja, Lawler, Sean E., Qu, Yuan, Fadzen, Colin M., Wolfe, Justin, Regan, Michael S., Pentelute, Bradley L., Agar, Nathalie Y. R., Cho, Choi-Fong
Published 2020

In-solution enrichment identifies peptide inhibitors of protein-protein interactions

by Touti, Faycal, Gates, Zachary P, Bandyopadhyay, Anupam, Lautrette, Guillaume, Pentelute, Bradley L.
Published 2020

Following Natures Lead: On the Construction of Membrane-Inserted Toxins in Lipid Bilayer Nanodiscs

by Akkaladevi, Narahari, Mukherjee, Srayanta, Katayama, Hiroo, Janowiak, Blythe, Patel, Deepa, Gogol, Edward P., Pentelute, Bradley L., John Collier, R., Fisher, Mark T.
Published 2017