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Ashfaq, U.A
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Ashfaq, U.A
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Ashfaq, U.A
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1
Discovery of amide-functionalized benzimidazolium salts as potent α-glucosidase inhibitors
by
Ahmad, M.
,
Ashfaq
,
U.A
,
Khan, I.A
,
Sultan, S.
,
Zaki, M.E.A
Published 2021
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2
Synthesis and α-glucosidase inhibition activity of 2-[3-(Benzoyl/4-bromobenzoyl)-4-hydroxy-1,1-dioxido-2h-benzo[e][1,2]thiazin-2-yl]-n-arylacetamides: An in silico and biochemical...
by
Ahmad, M.
,
Ashfaq
,
U.A
,
Aslam, S.
,
Hussain, M.
,
Lee, D.S
,
Muddassar, M.
,
Saddique, F.A
,
Sultan, S.
,
Taj, S.
,
Zaki, M.E.A
Published 2021
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Related Subjects
Glycoside Hydrolase Inhibitors
Molecular Docking Simulation
Molecular docking
Structure-Activity Relationship
chemistry
glycosidase inhibitor
molecular docking
structure activity relation
α-glucosidase inhibition
1,2-Benzothiazines
Acetamides
Amides
Anti-diabetic
Anti-diabetic studies
Benzimidazole derivatives
Benzimidazoles
Benzimidazolium salts
Catalytic Domain
Computer Simulation
Diabetes Mellitus
Drug Design
Drug Evaluation, Preclinical
Humans
Hypoglycemic Agents
IC50
Inhibitory Concentration 50
Kinetics
Salts
Synthesis
Thiazines
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