Allosteric Modulation of GPCRs of Class A by Cholesterol

by Jan Jakubík, Esam E. El-Fakahany
Published 2021-02-01

Allosteric Modulation of Muscarinic Acetylcholine Receptors

by Esam E. El-Fakahany, Jan Jakubík
Published 2010-08-01

Current Advances in Allosteric Modulation of Muscarinic Receptors

by Jan Jakubik, Esam E. El-Fakahany
Published 2020-02-01

Analysis of equilibrium binding of an orthosteric tracer and two allosteric modulators.

by Jan Jakubík, Alena Randáková, Esam E El-Fakahany, Vladimír Doležal
Published 2019-01-01

Long-term activation upon brief exposure to xanomleline is unique to M1 and M4 subtypes of muscarinic acetylcholine receptors.

by Eva Šantrůčková, Vladimír Doležal, Esam E El-Fakahany, Jan Jakubík
Published 2014-01-01

Subtype differences in pre-coupling of muscarinic acetylcholine receptors.

by Jan Jakubík, Helena Janíčková, Alena Randáková, Esam E El-Fakahany, Vladimír Doležal
Published 2011-01-01

Pharmacological evaluation of the long-term effects of xanomeline on the M(1) muscarinic acetylcholine receptor.

by Marianne K O Grant, Meredith J Noetzel, Kayla C De Lorme, Jan Jakubík, Vladimír Doležal, Esam E El-Fakahany
Published 2010-12-01