The first Pd-catalyzed Buchwald–Hartwig aminations at C-2 or C-4 in the estrone series

by Ildikó Bacsa, Dávid Szemerédi, János Wölfling, Gyula Schneider, Lilla Fekete, Erzsébet Mernyák
Published 2018-05-01

Synthesis of substituted 15β-alkoxy estrone derivatives and their cofactor-dependent inhibitory effect on 17β-HSD1

by Bianka Edina Herman, Anita Kiss, János Wölfling, Erzsébet Mernyák, Mihály Szécsi, Gyula Schneider
Published 2019-01-01

Electrophile- and Lewis acid-induced nitrone formation and 1,3-dpolar cycloaddition reactions in the 13α- and 13β-estrone series

by Erzsebet Mernyak, Judit Huber, Gabriella Benedek, Roland Pfoh, Stephan Rühl, Gyula Schneider, János Wölfling
Published 2010-09-01

Synthesis of novel 13α-estrone derivatives by Sonogashira coupling as potential 17β-HSD1 inhibitors

by Ildikó Bacsa, Rebeka Jójárt, János Wölfling, Gyula Schneider, Bianka Edina Herman, Mihály Szécsi, Erzsébet Mernyák
Published 2017-06-01

Efficient synthesis of novel A-ring-substituted 1,2,3-triazolylcholestane derivatives via catalytic azide-alkyne cycloaddition

by Zalán Kádár, Éva Frank, Gyula Schneider, Judit Molnár, István Zupkó, János Kóti, Bruno Schönecker, János Wölfling
Published 2012-01-01

Synthesis and In Vitro Antiproliferative Activity of Novel Androst-5-ene Triazolyl and Tetrazolyl Derivatives

by János Wölfling, Tibor Bartók, Éva Frank, Gyula Schneider, Judit Huber, István Zupkó, Dóra Kovács, Zalán Kádár
Published 2011-06-01

Synthesis and in Vitro Antiproliferative Evaluation of C-13 Epimers of Triazolyl-d-Secoestrone Alcohols: The First Potent 13α-d-Secoestrone Derivative

by Johanna Szabó, Nóra Jerkovics, Gyula Schneider, János Wölfling, Noémi Bózsity, Renáta Minorics, István Zupkó, Erzsébet Mernyák
Published 2016-05-01

Synthesis, Biological Evaluation and Docking Studies of 13-Epimeric 10-fluoro- and 10-Chloroestra-1,4-dien-3-ones as Potential Aromatase Inhibitors

by Rebeka Jójárt, Péter Traj, Édua Kovács, Ágnes Horváth, Gyula Schneider, Mihály Szécsi, Attila Pál, Gábor Paragi, Erzsébet Mernyák
Published 2019-05-01

Antiproliferative Properties of Newly Synthesized 19-Nortestosterone Analogs Without Substantial Androgenic Activity

by András Gyovai, Renáta Minorics, Anita Kiss, Erzsébet Mernyák, Gyula Schneider, András Szekeres, Erika Kerekes, Imre Ocsovszki, István Zupkó, István Zupkó
Published 2018-07-01

Synthesis and Biological Evaluation of Triazolyl 13α-Estrone–Nucleoside Bioconjugates

by Brigitta Bodnár, Erzsébet Mernyák, János Wölfling, Gyula Schneider, Bianka Edina Herman, Mihály Szécsi, Izabella Sinka, István Zupkó, Zoltán Kupihár, Lajos Kovács
Published 2016-09-01

Synthesis and structure–activity relationships of 2- and/or 4-halogenated 13β- and 13α-estrone derivatives as enzyme inhibitors of estrogen biosynthesis

by Ildikó Bacsa, Bianka Edina Herman, Rebeka Jójárt, Kevin Stefán Herman, János Wölfling, Gyula Schneider, Mónika Varga, Csaba Tömböly, Tea Lanišnik Rižner, Mihály Szécsi, Erzsébet Mernyák
Published 2018-01-01