The Efficacy of the Novel TSPO Ligands 2-Cl-MGV-1 and 2,4-Di-Cl-MGV-1 Compared to the Classical TSPO Ligand PK 11195 to Counteract the Release of Chemokines from LPS-Stimulated BV-...

by Sheelu Monga, Abraham Weizman, Moshe Gavish
Published 2020-09-01

Effects of Cigarette Smoke on TSPO-related Mitochondrial Processes

by Nidal Zeineh, Rafael Nagler, Martin Gabay, Abraham Weizman, Moshe Gavish
Published 2019-07-01

The TSPO Ligands 2-Cl-MGV-1, MGV-1, and PK11195 Differentially Suppress the Inflammatory Response of BV-2 Microglial Cell to LPS

by Maya Azrad, Nidal Zeineh, Abraham Weizman, Leo Veenman, Moshe Gavish
Published 2019-01-01

Inhibitory Effects of the Two Novel TSPO Ligands 2-Cl-MGV-1 and MGV-1 on LPS-induced Microglial Activation

by Sheelu Monga, Rafi Nagler, Rula Amara, Abraham Weizman, Moshe Gavish
Published 2019-05-01

Tetrapyrroles as Endogenous TSPO Ligands in Eukaryotes and Prokaryotes: Comparisons with Synthetic Ligands

by Leo Veenman, Alex Vainshtein, Nasra Yasin, Maya Azrad, Moshe Gavish
Published 2016-06-01

Efficaciousness of Low Affinity Compared to High Affinity TSPO Ligands in the Inhibition of Hypoxic Mitochondrial Cellular Damage Induced by Cobalt Chloride in Human Lung H1299 Cel...

by Nidal Zeineh, Nunzio Denora, Valentino Laquintana, Massimo Franco, Abraham Weizman, Moshe Gavish
Published 2020-05-01

Ligands of the Mitochondrial 18 kDa Translocator Protein Attenuate Apoptosis of Human Glioblastoma Cells Exposed to Erucylphosphohomocholine

by Wilfried Kugler, Leo Veenman, Yulia Shandalov, Svetlana Leschiner, Ilana Spanier, Max Lakomek, Moshe Gavish
Published 2008-01-01

The TSPO Ligands MGV-1 and 2-Cl-MGV-1 Differentially Inhibit the Cigarette Smoke-Induced Cytotoxicity to H1299 Lung Cancer Cells

by Nidal Zeineh, Rafael M. Nagler, Martin Gabay, Fadi Obeid, Meygal Kahana, Abraham Weizman, Moshe Gavish
Published 2021-05-01

The protective effect of the TSPO ligands 2,4-Di-Cl-MGV-1, CB86, and CB204 against LPS-induced M1 pro-inflammatory activation of microglia

by Sheelu Monga, Nunzio Denora, Valentino Laquintana, Massimo Franco, Ilan Marek, Sukhdev Singh, Rafi Nagler, Abraham Weizman, Moshe Gavish
Published 2020-05-01

Sunitinib-Containing Carborane Pharmacophore with the Ability to Inhibit Tyrosine Kinases Receptors FLT3, KIT and PDGFR-β, Exhibits Powerful In Vivo Anti-Glioblastoma Activity

by Catalina Alamón, Belén Dávila, María Fernanda García, Carina Sánchez, Mariángeles Kovacs, Emiliano Trias, Luis Barbeito, Martín Gabay, Nidal Zeineh, Moshe Gavish, Francesc Teixidor, Clara Viñas, Marcos Couto, Hugo Cerecetto
Published 2020-11-01