Prodrug Strategy in Drug Development

Prodrugs are chemically modified derivatives introduced in therapy due to their advantageous physico-chemical properties (greater stability, improved solubility, increased permeability), used in inactive form. Biological effect is exerted by the active derivatives formed in organism through chemical...

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Bibliographic Details
Main Authors: Hajnal Kelemen, Gabriel Hancu, Aura Rusu, Erzsébet Varga, Blanka Székely Szentmiklósi
Format: Article
Language:English
Published: Sciendo 2016-09-01
Series:Acta Medica Marisiensis
Subjects:
Online Access:https://doi.org/10.1515/amma-2016-0032