The synthesis and preliminary pharmacological evaluation of the racemic cis and trans 3-alkylfentanyl analogues
A general, five step method for the synthesis of 3-alkylfentanyl analogues (i.e., cis and trans 3-alkyl-4-anilidopiperidines 6.16.6) has been developed. The starting N-phenethyl-4-piperidone 1 was first converted into the cyclohexylimine derivative 2, a-deprotonated with butyllithium and the resulti...
| Main Authors: | , , , , , , , |
|---|---|
| Format: | Article |
| Language: | English |
| Published: |
Serbian Chemical Society
2004-07-01
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| Series: | Journal of the Serbian Chemical Society |
| Online Access: | http://www.shd.org.yu/HtDocs/SHD/Vol69/No7/V69-No7-01.pdf |