Study on Biopharmaceutics Classification and Oral Bioavailability of a Novel Multikinase Inhibitor NCE for Cancer Therapy

Specific biopharmaceutics classification investigation and study on phamacokinetic profile of a novel drug candidate (2-methylcarbamoyl-4-{4-[3- (trifluoromethyl) benzamido] phenoxy} pyridinium 4-methylbenzenesulfonate monohydrate, NCE) were carried out. Equilibrium solubility and intrinsic dissolut...

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Bibliographic Details
Main Authors: Yang Yang, Chun-Mei Fan, Xuan He, Ke Ren, Jin-Kun Zhang, Ying-Ju He, Luo-Ting Yu, Ying-Lan Zhao, Chang-Yang Gong, Yu Zheng, Xiang-Rong Song, Jun Zeng
Format: Article
Language:English
Published: MDPI AG 2014-04-01
Series:International Journal of Molecular Sciences
Subjects:
Online Access:http://www.mdpi.com/1422-0067/15/5/7199