Design, Radiosynthesis and Preliminary Biological Evaluation in Mice of a Brain-Penetrant <sup>18</sup>F-Labelled σ<sub>2</sub> Receptor Ligand
The σ<sub>2</sub> receptor (transmembrane protein 97), which is involved in cholesterol homeostasis, is of high relevance for neoplastic processes. The upregulated expression of σ<sub>2</sub> receptors in cancer cells and tissue in combination with the antiproliferative poten...
Main Authors: | Rareş-Petru Moldovan, Daniel Gündel, Rodrigo Teodoro, Friedrich-Alexander Ludwig, Steffen Fischer, Magali Toussaint, Dirk Schepmann, Bernhard Wünsch, Peter Brust, Winnie Deuther-Conrad |
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Format: | Article |
Language: | English |
Published: |
MDPI AG
2021-05-01
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Series: | International Journal of Molecular Sciences |
Subjects: | |
Online Access: | https://www.mdpi.com/1422-0067/22/11/5447 |
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