Allosteric modulation of adenosine A1 and cannabinoid 1 receptor signaling by G‐peptides

Abstract While allosteric modulation of GPCR signaling has gained prominence to address the need for receptor specificity, efforts have mainly focused on allosteric sites adjacent to the orthosteric ligand‐binding pocket and lipophilic molecules that target transmembrane helices. In this study, we e...

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Bibliographic Details
Main Authors: Anja M. Touma, Rabia U. Malik, Tejas Gupte, Sivaraj Sivaramakrishnan
Format: Article
Language:English
Published: Wiley 2020-12-01
Series:Pharmacology Research & Perspectives
Subjects:
Online Access:https://doi.org/10.1002/prp2.673