C4-Alkylamination of C4-Halo-1<i>H</i>-1-tritylpyrazoles Using Pd(dba)<sub>2</sub> or CuI

Alkylamino coupling reactions at the C4 positions of 4-halo-1<i>H</i>-1-tritylpyrazoles were investigated using palladium or copper catalysts. The Pd(dba)<sub>2</sub> catalyzed C-N coupling reaction of aryl- or alkylamines, lacking a β-hydrogen atom, proceeded smoothly using...

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Bibliographic Details
Main Authors: Yoshihide Usami, Yuya Tatsui, Hiroki Yoneyama, Shinya Harusawa
Format: Article
Language:English
Published: MDPI AG 2020-10-01
Series:Molecules
Subjects:
Online Access:https://www.mdpi.com/1420-3049/25/20/4634