Optimized Structure-based Methodology for Studying PPARγ Partial Agonists

The peroxisome proliferator-activated receptor (PPAR) γ is a master regulator of the lipid and glucose metabolism, and thus is a valuable drug target. Since its full activation is accompanied by a number of adverse effects, researchers focus on discovery of novel compounds with ligand-receptor inter...

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Bibliographic Details
Main Authors: Merilin Al Sharif, Antonia Diukendjieva, Petko Alov, Ivanka Tsakovska, Ilza Pajeva
Format: Article
Language:English
Published: Bulgarian Academy of Sciences 2018-03-01
Series:International Journal Bioautomation
Subjects:
Online Access:http://www.biomed.bas.bg/bioautomation/2018/vol_22.1/files/22.1_07.pdf