Synthesis, antibacterial activities, and sustained perfume release properties of optically active5-hydroxy- and 5-acetoxyalkanethioamide analogues

5-Acetoxy- and 5-hydroxyalkanethioamide analogues showed high antibacterial activity against Staphylococcus aureus. Antibacterial thioamides were prepared from 5-alkyl-δ-lactones by amidation, thionation, and subsequent deacetylation. Optically active thioamides with 99% diastereomeric excesses were...

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Bibliographic Details
Main Authors: Shimotori Yasutaka, Hoshi Masayuki, Ogawa Narihito, Miyakoshi Tetsuo, Kanamoto Taisei
Format: Article
Language:English
Published: De Gruyter 2020-06-01
Series:Heterocyclic Communications
Subjects:
Online Access:http://www.degruyter.com/view/j/hc.2020.26.issue-1/hc-2019-0103/hc-2019-0103.xml?format=INT