C7-Derivatization of C3-Alkylindoles Including Tryptophans and Tryptamines

C7-Derivatization of C3-Alkylindoles Including Tryptophans and Tryptamines

A versatile strategy for C7-selective boronation of tryptophans, tryptamines, and 3-alkylindoles by way of a single-pot C2/C7-diboronation-C2-protodeboronation sequence is described. The combination of a mild iridium-catalyzed C2/C7-diboronation followed by an in situ palladium-catalyzed C2-protodeb...

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Bibliographic Details
Main Authors: Loach, Richard Peter (Contributor), Fenton, Owen S. (Contributor), Amaike, Kazuma (Contributor), Siegel, Dustin Scott (Contributor), Ozkal, Erhan (Contributor), Movassaghi, Mohammad (Contributor)
Other Authors: Massachusetts Institute of Technology. Department of Chemistry (Contributor)
Format: Article
Language:English
Published: American Chemical Society (ACS), 2017-06-09T19:58:33Z.
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