C7-Derivatization of C3-Alkylindoles Including Tryptophans and Tryptamines
A versatile strategy for C7-selective boronation of tryptophans, tryptamines, and 3-alkylindoles by way of a single-pot C2/C7-diboronation-C2-protodeboronation sequence is described. The combination of a mild iridium-catalyzed C2/C7-diboronation followed by an in situ palladium-catalyzed C2-protodeb...
Main Authors: | , , , , , |
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Format: | Article |
Language: | English |
Published: |
American Chemical Society (ACS),
2017-06-09T19:58:33Z.
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Subjects: | |
Online Access: | Get fulltext |