Regioselective Synthesis of Benzimidazolones via Cascade C-N Coupling of Monosubstituted Ureas

A direct method for the regioselective construction of benzimidazolones is reported wherein a single palladium catalyst is employed to couple monosubstituted urea substrates with differentially substituted 1,2-dihaloaromatic systems. In this method, the catalyst is able to promote a cascade of two d...

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Bibliographic Details
Main Authors: Ernst, Johannes B. (Contributor), Tay, Nicholas E. S. (Contributor), Jui, Nathan T. (Contributor), Buchwald, Stephen Leffler (Contributor)
Other Authors: Massachusetts Institute of Technology. Department of Chemistry (Contributor)
Format: Article
Language:English
Published: American Chemical Society (ACS), 2015-11-03T12:44:13Z.
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