New methodologies for thioacylation of amines and thiopeptides synthesis
The synthesis of an analog of Leucine enkephalin bearing a thioamide linkage in position 3 was accomplished. Attempts to couple thiodipeptides to amines by the means of activating their free carboxyl function was showed to give substituted thiazolones which were not found suitable for the synthesis...
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| Format: | Others |
| Language: | en |
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McGill University
1985
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| Online Access: | http://digitool.Library.McGill.CA:80/R/?func=dbin-jump-full&object_id=71997 |