Inhibitory Effects of Quercetin and Its Main Methyl, Sulfate, and Glucuronic Acid Conjugates on Cytochrome P450 Enzymes, and on OATP, BCRP and MRP2 Transporters

Quercetin is a flavonoid, its glycosides and aglycone are found in significant amounts in several plants and dietary supplements. Because of the high presystemic biotransformation of quercetin, mainly its conjugates appear in circulation. As has been reported in previous studies, quercetin can inter...

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Bibliographic Details
Main Authors: Violetta Mohos, Eszter Fliszár-Nyúl, Orsolya Ungvári, Katalin Kuffa, Paul W. Needs, Paul A. Kroon, Ágnes Telbisz, Csilla Özvegy-Laczka, Miklós Poór
Format: Article
Language:English
Published: MDPI AG 2020-07-01
Series:Nutrients
Subjects:
Online Access:https://www.mdpi.com/2072-6643/12/8/2306