FLUOROUS SUPPORTED SYNTHESIS OF PYRAZOLONE DERIVATIVES FROM ALLYLIC ALCOHOLS USING A PALLADIUM-CATALYZED STRATEGY

Ten substituted pyrazolone derivatives were easily synthesized from perfluorinated allylic alcohols, via a straightforward two steps reaction involving a Heck-coupling/isomerization reaction and subsequent condensation of hydrazines. This fluorous supported methodology, that combines a cyclo-release...

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Bibliographic Details
Main Authors: Nicolas Gouault, Alexandre Cariou, Jean-François Cupif, Patrícia de Aguiar Amaral, Michèle David
Format: Article
Language:English
Published: Sociedade Brasileira de Química
Series:Química Nova
Subjects:
Online Access:http://www.scielo.br/scielo.php?script=sci_arttext&pid=S0100-40422016000700825&lng=en&tlng=en