Synthesis and in Vitro Antiproliferative Evaluation of C-13 Epimers of Triazolyl-d-Secoestrone Alcohols: The First Potent 13α-d-Secoestrone Derivative

by Johanna Szabó, Nóra Jerkovics, Gyula Schneider, János Wölfling, Noémi Bózsity, Renáta Minorics, István Zupkó, Erzsébet Mernyák
Published 2016-05-01

Sequential Ugi reaction/base-induced ring closing/IAAC protocol toward triazolobenzodiazepine-fused diketopiperazines and hydantoins

by Robby Vroemans, Fante Bamba, Jonas Winters, Joice Thomas, Jeroen Jacobs, Luc Van Meervelt, Jubi John, Wim Dehaen
Published 2018-03-01

Efficient catenane synthesis by cucurbit[6]uril-mediated azide–alkyne cycloaddition

by Antony Wing Hung Ng, Chi-Chung Yee, Kai Wang, Ho Yu Au-Yeung
Published 2018-07-01

Synthesis and evaluation of anticancer activities of 2- or 4-substituted 3-(N-benzyltriazolylmethyl)-13α-oestrone derivatives

by Rebeka Jójárt, Seyyed Ashkan Senobar Tahaei, Péter Trungel-Nagy, Zoltán Kele, Renáta Minorics, Gábor Paragi, István Zupkó, Erzsébet Mernyák
Published 2021-01-01

Combination of Photoinduced ATRP and Click Processes for the Synthesis of Triblock Copolymers

by Görkem Yılmaz
Published 2018-01-01

Copper(I)-Catalyzed Click Chemistry as a Tool for the Functionalization of Nanomaterials and the Preparation of Electrochemical (Bio)Sensors

by P. Yáñez-Sedeño, A. González-Cortés, S. Campuzano, J. M. Pingarrón
Published 2019-05-01

Stepwise, Protecting Group Free Synthesis of [4]Rotaxanes

by James E. M. Lewis, Joby Winn, Stephen M. Goldup
Published 2017-01-01

Ion-Conducting Redox-Active Polymer Gels Based on Stable Nitroxide Radicals

by Fadoi Boujioui, Jean-François Gohy
Published 2019-08-01

Design and Synthesis of Various 5′-Deoxy-5′-(4-Substituted-1,2,3-Triazol-1-yl)-Uridine Analogues as Inhibitors of <i>Mycobacterium tuberculosis</i> Mur Ligases

by Vincent Hervin, Ritu Arora, Jyoti Rani, Srinivasan Ramchandran, Urmi Bajpai, Luigi A. Agrofoglio, Vincent Roy
Published 2020-10-01

Phenylglyoxal-Based Visualization of Citrullinated Proteins on Western Blots

by Sanne M. M. Hensen, Wilbert C. Boelens, Kimberly M. Bonger, Remco T. P. van Cruchten, Floris L. van Delft, Ger J. M. Pruijn
Published 2015-04-01

Synthetic Strategy and Anti-Tumor Activities of Macrocyclic Scaffolds Based on 4-Hydroxyproline

by Guorui Cao, Kun Yang, Yue Li, Longjiang Huang, Dawei Teng
Published 2016-02-01

Modified Nucleosides, Nucleotides and Nucleic Acids via Click Azide-Alkyne Cycloaddition for Pharmacological Applications

by Daniela Perrone, Elena Marchesi, Lorenzo Preti, Maria Luisa Navacchia
Published 2021-05-01

Micellar Carriers Based on Amphiphilic PEG/PCL Graft Copolymers for Delivery of Active Substances

by Justyna Odrobińska, Dorota Neugebauer
Published 2020-11-01

A highly sensitive protocol for microscopy of alkyne lipids and fluorescently tagged or immunostained proteins[S]

by Anne Gaebler, Anke Penno, Lars Kuerschner, Christoph Thiele
Published 2016-10-01

Synthesis of (1,2,3-triazol-4-yl)methyl Phosphinates and (1,2,3-Triazol-4-yl)methyl Phosphates by Copper-Catalyzed Azide-Alkyne Cycloaddition

by Anna Tripolszky, Krisztina Németh, Pál Tamás Szabó, Erika Bálint
Published 2019-05-01

Designed Artificial Protein Heterodimers With Coupled Functions Constructed Using Bio-Orthogonal Chemistry

by Rachel L. Johnson, Hayley G. Blaber, Hayley G. Blaber, Tomas Evans, Harley L. Worthy, Harley L. Worthy, Jacob R. Pope, D. Dafydd Jones
Published 2021-08-01

Increasing Polarity in Tacrine and Huprine Derivatives: Potent Anticholinesterase Agents for the Treatment of Myasthenia Gravis

by Carles Galdeano, Nicolas Coquelle, Monika Cieslikiewicz-Bouet, Manuela Bartolini, Belén Pérez, M. Victòria Clos, Israel Silman, Ludovic Jean, Jacques-Philippe Colletier, Pierre-Yves Renard, Diego Muñoz-Torrero
Published 2018-03-01

Design and Synthesis of New 5-aryl-4-Arylethynyl-1<i>H</i>-1,2,3-triazoles with Valuable Photophysical and Biological Properties

by Mariia M. Efremova, Anastasia I. Govdi, Valeria V. Frolova, Andrey M. Rumyantsev, Irina A. Balova
Published 2021-05-01

Synthesis and Antiviral Evaluation of (1,4-Disubstituted-1,2,3-Triazol)-<i>(E)</i>-2-Methyl-but-2-Enyl Nucleoside Phosphonate Prodrugs

by Tuniyazi Abuduaini, Vincent Roy, Julien Marlet, Catherine Gaudy-Graffin, Denys Brand, Cécile Baronti, Franck Touret, Bruno Coutard, Tamara R. McBrayer, Raymond F. Schinazi, Luigi A. Agrofoglio
Published 2021-03-01

Synthesis of a New Polyanion Possessing Dense 1,2,3-Triazole Backbone

by Linlin Xu, Yuri Kamon, Akihito Hashidzume
Published 2021-05-01